• Title of article

    Design and synthesis of sulfonyl-substituted 4,5-diarylthiazoles as selective cyclooxygenase-2 inhibitors

  • Author/Authors

    Jeffery S. Carter، نويسنده , , D. J. Rogier، نويسنده , , Matthew J. Graneto، نويسنده , , Karen Seibert and، نويسنده , , Carol M. Koboldt، نويسنده , , Yan Zhang، نويسنده , , John J. Talley، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    4
  • From page
    1167
  • To page
    1170
  • Abstract
    A series of novel sulfone substituted 4,5-diarylthiazoles have been synthesized and evaluated for their inhibition of the two isoforms of human cyclooxygenase (COX-1 and COX-2). This series displays exceptionally selective COX-2 inhibition.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1999
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790112