• Title of article

    Synthesis and in vitro and in vivo evaluation of the 2-(6′methoxy-3′,4′-dihydro-1′-naphtyl)-4H-3,1-benzoxazin-4-one as a new potent substrate inhibitor of human leukocyte elastase

  • Author/Authors

    Antonio Arcadi، نويسنده , , Cinzia Asti، نويسنده , , Laura Brandolini، نويسنده , , Gianfranco Caselli، نويسنده , , Fabio Marinelli، نويسنده , , Viviana Ruggieri، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    4
  • From page
    1291
  • To page
    1294
  • Abstract
    the title 2-vinyl-4H-3,1-benzoxazin-4-one has been synthesised and tested for inhibitory activity against human leukocyte elastase. The compound has shown activity both in vitro towards human sputum elastase and in vivo in an hemorrhagic assay.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1999
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790137