• Title of article

    C32-O-phenalkyl ether derivatives of the immunosuppressant ascomycin: a tether length study

  • Author/Authors

    Mark T. Goulet، نويسنده , , Peter J. Sinclair، نويسنده , , Frederick Wong، نويسنده , , Mary Jo Staruch، نويسنده , , Francis J. Dumont، نويسنده , , John G. Cryan، نويسنده , , Gregory J. Wiederrecht، نويسنده , , Matthew J. Wyvratt Jr.، نويسنده , , William H. Parsons، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    4
  • From page
    2085
  • To page
    2088
  • Abstract
    A tether length study of C32-O-phenalkyl ether derivatives of ascomycin was conducted wherein it was determined that a 2-carbon tether provides optimum in vitro immunosuppressive activity. Oxygen-bearing substituents along the 2-carbon tether can further increase the potency of this design.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1999
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790289