• Title of article

    Dysidiolide and related γ-hydroxy butenolide compounds as inhibitors of the protein tyrosine phosphatase, CDC25

  • Author/Authors

    Jill L. Blanchard، نويسنده , , David M. Epstein، نويسنده , , Michael D. Boisclair، نويسنده , , Johannes Rudolph، نويسنده , , Kollol Pal، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    2
  • From page
    2537
  • To page
    2538
  • Abstract
    Synthetic dysidiolide, as well as several related compounds containing a γ-hydroxybutenolide moiety, were tested in in vitro Cdc25 assays against both synthetic and natural substrates. Contrary to literature values which are in the low micromolar range, we observe only millimolar inhibitory activity for these compounds versus Cdc25 phosphatase.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    1999
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790381