Title of article
Delta opioid binding selectivity of 3-ether analogs of naltrindole
Author/Authors
Andrew Coop، نويسنده , , Julia Pinto، نويسنده , , Lijuan Wang، نويسنده , , Karen McCullough، نويسنده , , Richard B. Rothman، نويسنده , , Christine Dersch، نويسنده , , Arthur E. Jacobson، نويسنده , , Kenner C. Rice، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 1999
Pages
4
From page
3435
To page
3438
Abstract
Masking of the 3-phenol of naltrindole as a range of ethers caused a decrease in binding affinity at all three opiate receptors (μ, κ, δ), however for the methyl ether, the reduction in affinity at both μ and κ was greater than at δ, thereby increasing δ binding selectivity.
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
1999
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
790550
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