• Title of article

    Recognition and inhibition of HIV integrase by a novel dinucleotide

  • Author/Authors

    Michael Taktakishvili، نويسنده , , Nouri Neamati، نويسنده , , Yves Pommier، نويسنده , , Vasu Nair، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2000
  • Pages
    3
  • From page
    249
  • To page
    251
  • Abstract
    The viral enzyme, HIV integrase, is involved in the integration of viral DNA into host cell DNA. In the quest for a small nucleotide system with nuclease stability of the internucleotide phosphate bond and critical structural features for recognition and inhibition of HIV-1 integrase, we have discovered a conceptually novel dinucleotide, pIsodApdC, which is a potent inhibitor of this key viral enzyme.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2000
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    790614