Title of article
Furans with basic side chains: synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha
Author/Authors
Deborah S. Mortensen، نويسنده , , Alice L. Rodriguez، نويسنده , , Jun Sun، نويسنده , , Benita S. Katzenellenbogen، نويسنده , , John A. Katzenellenbogen، نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2001
Pages
4
From page
2521
To page
2524
Abstract
3-Alkyl-2,4,5-triarylfurans with basic side-chain substituents were prepared as ligands for the estrogen receptor. Those analogues having the basic side chain on the C(4) phenol were high-affinity, ERα-selective antagonists.
Journal title
Bioorganic & Medicinal Chemistry Letters
Serial Year
2001
Journal title
Bioorganic & Medicinal Chemistry Letters
Record number
791670
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