• Title of article

    Solid-phase synthesis of c(RGDfK) derivatives: on-resin cyclisation and lysine functionalisation

  • Author/Authors

    Catherine F. McCusker، نويسنده , , Philip J. Kocienski، نويسنده , , F. Thomas Boyle، نويسنده , , Andreas G. Sch?tzlein، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2002
  • Pages
    3
  • From page
    547
  • To page
    549
  • Abstract
    The cyclic pentapeptide c(RGDfK), a selective ligand for the αvβ3 integrin, was synthesised on solid phase. All synthetic operations including the cyclisation step and the appendage of the Bolton–Hunter reagent was conducted on-resin.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2002
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    792015