• Title of article

    Peptidomimetics of Efflux Pump Inhibitors Potentiate the Activity of Levofloxacin in Pseudomonas aeruginosa

  • Author/Authors

    Thomas E. Renau، نويسنده , , Roger Léger، نويسنده , , Rose Yen، نويسنده , , Miles W. She، نويسنده , , Eric M. Flamme، نويسنده , , Joan Sangalang، نويسنده , , Carla L. Gannon، نويسنده , , Suzanne Chamberland، نويسنده , , Olga Lomovskaya، نويسنده , , Ving J. Lee، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2002
  • Pages
    4
  • From page
    763
  • To page
    766
  • Abstract
    Several classes of peptidomimetics of the efflux pump inhibitor -ornithine- -homophenylalanine-3-aminoquinoline (MC-02,595) have been prepared and evaluated for their ability to potentiate the activity of the fluoroquinolone levofloxacin in Pseudomonas aeruginosa. A number of the new analogues were as active or more active than the lead, demonstrating that a peptide backbone is not essential for activity.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2002
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    792063