• Title of article

    Antibacterial activity of G6-quaternary ammonium derivatives of a lipophilic vancomycin analogue

  • Author/Authors

    Timothy A. Blizzard، نويسنده , , Ronald M. Kim، نويسنده , , Jerry D. Morgan، نويسنده , , II، نويسنده , , Sheng-Jiang Chang، نويسنده , , Joyce Kohler، نويسنده , , Ruth Kilburn، نويسنده , , Kevin Chapman، نويسنده , , Milton L. Hammond، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2002
  • Pages
    4
  • From page
    849
  • To page
    852
  • Abstract
    A series of G6-amino derivatives of a lipophilic vancomycin analogue was prepared. Antibacterial activity of the analogues was inversely proportional to the degree of substitution of the G6-nitrogen. The fully substituted (quaternary) analogues were essentially inactive against vanA phenotype VREF strains but retained substantial activity against other bacteria, a profile reminiscent of teicoplanin.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2002
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    792083