• Title of article

    Novel Inhibitors of Plasminogen Activator Inhibitor-1: Development of New Templates From Diketopiperazines

  • Author/Authors

    Shouming Wang، نويسنده , , Julian Golec، نويسنده , , Warren Miller، نويسنده , , Sandra Milutinovic، نويسنده , , Adrian Folkes، نويسنده , , Susannah Williams، نويسنده , , Teresa Brooks، نويسنده , , Kevin Hardman، نويسنده , , Peter Charlton، نويسنده , , Stephen Wren، نويسنده , , John Spencer، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2002
  • Pages
    4
  • From page
    2367
  • To page
    2370
  • Abstract
    Several isoquinoline-based templates were identified from the studies of the conformational effects of the diketopiperazine structures for PAI-1 inhibition. Moderate to good activity was retained with the elimination of unattractive characteristics in the diketopiperazine template.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2002
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    792449