• Title of article

    Pyrimidinone antibiotics—heterocyclic analogues with improved antibacterial spectrum

  • Author/Authors

    Michael Brands، نويسنده , , Yolanda Cancho Grande، نويسنده , , Rainer Endermann، نويسنده , , Reinhold Gahlmann، نويسنده , , Jochen Krüger، نويسنده , , Siegfried Raddatz، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2003
  • Pages
    5
  • From page
    2641
  • To page
    2645
  • Abstract
    We report the synthesis and pharmacological evaluation of new derivatives of the natural dipeptide antibiotic TAN 1057 A,B containing heterocycles either in the β-amino acid side chain or as mimics of the urea function. In the course of this program, we identified novel analogues that display activity towards a broader panel of Gram-positive bacteriae.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2003
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    793417