• Title of article

    Ganglioside GM1 mimics: lipophilic substituents improve affinity for cholera toxin

  • Author/Authors

    Daniela Arosio، نويسنده , , Sergio Baretti، نويسنده , , Stefania Cattaldo، نويسنده , , Donatella Potenza، نويسنده , , Anna Bernardi، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2003
  • Pages
    4
  • From page
    3831
  • To page
    3834
  • Abstract
    Ganglioside GM1 mimics including (R)-2-hydroxy-3-cyclohexylpropionic acid or (R)-2-hydroxy-3-phenylpropionic acid as replacements for NeuAc are stronger cholera toxin binders than the parent ligand 2, which includes (R)-2-hydroxy-propionic acid.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2003
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    793668