• Title of article

    Fluorinated quinoid inhibitor: possible `pureʹ arylator predicted by the simple theoretical calculation

  • Author/Authors

    Seung Wook Ham، نويسنده , , Jong-In Choe، نويسنده , , Meifang Wang، نويسنده , , Vincent Peyregne، نويسنده , , Brian I Carr، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2004
  • Pages
    3
  • From page
    4103
  • To page
    4105
  • Abstract
    We report on the fluorinated form of Cpd 5 as a cell growth inhibitor. This compound is 3-fold more potent than the parent Cpd 5 and is predicted, using the semi-empirical AM1 method to be only an arylator of cysteine-containing proteins, without generating reactive oxygen species.
  • Keywords
    Reduction potential.* Corresponding author. Tel.: +1-412-624-6684 , fax: +1-412-624-6666 , Cdc25 inhibitor , e-mail: carrbi@msx.upmc.edu , Quinones
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2004
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    794744