• Title of article

    Synthesis and biological evaluation of DNA targeting flexible side-chain substituted β-carboline derivatives

  • Author/Authors

    Sulong Xiao، نويسنده , , Wei Lin، نويسنده , , Chao Wang، نويسنده , , Ming Yang، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2001
  • Pages
    5
  • From page
    437
  • To page
    441
  • Abstract
    A series of 3-substituted-β-carboline derivatives was synthesized from -tryptophan. The intercalating binding mode of these compounds with DNA, the effects of the flexible alkylamine side chain on the intercalating ability and their antitumor activity were studied, which agreed well with the molecular modeling results.
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Serial Year
    2001
  • Journal title
    Bioorganic & Medicinal Chemistry Letters
  • Record number

    800366