Title of article
Aziridination of Chiral 3-(2,2-Dimethyl-1,3-dioxolan-4-yl)-2-propenoate Esters
Author/Authors
Antonello Fazio، نويسنده , , M.Antonietta Loreto، نويسنده , , Paolo A Tardella، نويسنده , , Daniela Tofani، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2000
Pages
5
From page
4515
To page
4519
Abstract
The reactions of chiral 3-(2,2-dimethyl-1,3-dioxolan-4-yl)-2-propenoate esters 2–5 with NsONHCO2Et and CaO, produce the aziridine derivatives by addition of (ethoxycarbonyl)amino group on the double bond. The stereoselectivity is good for trans substrates. Products are precursors to polyhydroxy amino acids.
Keywords
Amination , Aziridines , amino acid derivatives , Esters
Journal title
Tetrahedron
Serial Year
2000
Journal title
Tetrahedron
Record number
1080942
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