Title of article :
Pseudoaxially Disubstituted Cyclo-β3-tetrapeptide Scaffolds
Author/Authors :
Peter W. Sutton، نويسنده , , Adrian Bradley، نويسنده , , Jaume Farràs، نويسنده , , Pedro Romea، نويسنده , , Fèlix Urp?́، نويسنده , , Jaume Vilarrasa، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2000
Abstract :
An N,N-disubstituted cyclo-β3-tetrapeptide, identified as a potential molecular scaffold, has been synthesised on a multigram scale from β-homophenylalanine by employing a nosylate-based protection strategy. C2-Symmetric derivatives containing pseudoaxial, combinatorially addressable functionalities have been prepared from the parent cyclopeptide.
Keywords :
amino acids and derivatives , ?3-peptides , Sulfonamides , Macrocycles , Aziridines
Journal title :
Tetrahedron
Journal title :
Tetrahedron
