Intramolecular trapping of amides by 1-lithio-1-bromocyclopropanes
Author/Authors :
Mark S Baird، نويسنده , , Florian A.M. Huber، نويسنده , , Viacheslav V. Tverezovsky، نويسنده , , Ivan G. Bolesov، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2001
Pages :
8
From page :
1593
To page :
1600
Abstract :
Reaction of 2-acylaminomethyl-1,1-dibromocyclopropanes with methyllithium at −90°C leads to selective bromine-lithium exchange and cyclisation to give a 1-bromo-3-azabicyclo[3.1.0]hexan-2-ol.