• Title of article

    Moenomycin analogues with modified lipid side chains from indium-mediated Barbier-type reactions

  • Author/Authors

    Stefan Vogel، نويسنده , , Katherina Stembera، نويسنده , , Lothar Hennig، نويسنده , , Matthias Findeisen، نويسنده , , Sabine Giesa، نويسنده , , Peter Welzel، نويسنده , , Maxime Lampilas*، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    8
  • From page
    4139
  • To page
    4146
  • Abstract
    From moenomycin A both the chromophore part and the lipid side chain were degraded by ozonolysis to give an analogue with a glycolaldehyde unit in 2-position of the glyceric acid moiety. The aldehyde was converted to a number of homoallylic alcohols by indium-mediated Barbier-type reactions with allylic and benzylic halides. With exception of the phytyl bromide-derived reaction product all compounds were antibiotically inactive.
  • Keywords
    Barbier reactions , Phospholipids , Carbohydrates , Antibiotics
  • Journal title
    Tetrahedron
  • Serial Year
    2001
  • Journal title
    Tetrahedron
  • Record number

    1082002