• Title of article

    A convenient synthesis of 3,4-difunctionalized δ-carbolines

  • Author/Authors

    Cyril Papamicaël، نويسنده , , Guy Queguiner، نويسنده , , Jean Bourguignon، نويسنده , , Georges Dupas، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2001
  • Pages
    7
  • From page
    5385
  • To page
    5391
  • Abstract
    An efficient and direct preparation of functionalized δ-carbolines, via a ring closure reaction between the appropriate indole amine and a masked 1,3-dicarbonyl compound is described. This method afforded new 3-substituted δ-carbolines and these products were subjected to ortho-lithiation experiments. Various 3,4-disubstituted δ-carbolines were obtained in acceptable yields.
  • Keywords
    Indoles , Cyclization , polycyclic heterocyclic compounds , Nitrogen heterocycles , lithiation , regioselection , Polycyclic aromatic compounds
  • Journal title
    Tetrahedron
  • Serial Year
    2001
  • Journal title
    Tetrahedron
  • Record number

    1082132