Title of article
Palladium-catalyzed direct arylation of thiazoles with aryl bromides
Author/Authors
Aya Yokooji، نويسنده , , Toru Okazawa، نويسنده , , Tetsuya Satoh، نويسنده , , Masahiro Miura، نويسنده , , Masakatsu Nomura، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2003
Pages
5
From page
5685
To page
5689
Abstract
Thiazole, 2-phenyl or -alkyl substituted one and benzothiazole are efficiently arylated with aryl bromides at the 2- and/or 5-position(s) in the presence of Pd(OAc)2 and a bulky phosphine ligand using Cs2CO3 as base. 2-Phenyl-5-thiazolecarboxanilide undergoes successive diarylation at the 4- and 5-positions accompanied by decarbamoylation.
Keywords
palladium and compounds , aryl halides , Thiazoles , arylation
Journal title
Tetrahedron
Serial Year
2003
Journal title
Tetrahedron
Record number
1088049
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