Title of article :
Palladium(II)-catalyzed heterocyclisation of 8-arylethynyl-1,2,3,4-tetrahydroquinolines: a facile route to 2-aryl-5,6-dihydro-4H-pyrrolo[3,2,1-ij]quinoline derivatives
Author/Authors :
Pascal Marchand، نويسنده , , Alain Puget، نويسنده , , Guillaume Le Baut، نويسنده , , Peter Emig، نويسنده , , Michael Czech، نويسنده , , Eckhard Günther، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2005
Abstract :
Dihydropyrroloquinolines have been synthesized reacting 8-arylethynyl-1,2,3,4-tetrahydroquinolines in the presence of palladium(II) chloride catalyst. Heteroannulation has been achieved in good yields and tolerates substituents on the tetrahydroquinoline, including bromo, cyano, and ester.
Keywords :
1-ij]quinolines , 3 , 4-Tetrahydroquinolines , 2 , 1 , Palladium(II)-catalyzed intramolecular heterocyclisation , 2 , 5
Journal title :
Tetrahedron
Journal title :
Tetrahedron
