• Title of article

    Efficient synthesis of cephalotaxine- and deoxyharringtonine analogues by a trimethylaluminium-mediated domino reaction

  • Author/Authors

    Lutz F. Tietze، نويسنده , , Holger Braun، نويسنده , , Peter L. Steck، نويسنده , , Serry A.A. El Bialy، نويسنده , , Nina T?lle، نويسنده , , Alexander Düfert، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2007
  • Pages
    9
  • From page
    6437
  • To page
    6445
  • Abstract
    The synthesis of cephalotaxine- and cephalotaxine amide analogues 14a–c and 16a–c as well as of the deoxyharringtonine analogues 5a,b was performed employing a trimethylaluminium-mediated domino reaction of 9a–c and 8 to give the spirocyclic compounds 7a–c, which was followed by a palladium catalyzed α-arylation.
  • Keywords
    Palladium , domino reactions , Alkaloids , Spiro compounds , Harringtonines , cephalotaxine
  • Journal title
    Tetrahedron
  • Serial Year
    2007
  • Journal title
    Tetrahedron
  • Record number

    1091121