Title of article
Solution-phase synthesis of 2-cyano and 2-amido aziridinyl peptides
Author/Authors
Stefania Fioravanti، نويسنده , , Davide Massari، نويسنده , , Alberto Morreale، نويسنده , , Lucio Pellacani، نويسنده , , Paolo A. Tardella، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2008
Pages
8
From page
3204
To page
3211
Abstract
Starting from a library of 2-l-α-amino acyl (E)-acrylonitriles, different short 2-cyano and 2-amido aziridinyl peptides, potential protease inhibitors, were obtained under parallel solution-phase conditions. The transformations include careful selection of conditions for aziridine deprotection and cyano group partial hydrolysis.
Journal title
Tetrahedron
Serial Year
2008
Journal title
Tetrahedron
Record number
1093921
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