• Title of article

    Developing an efficient route to the synthesis of nucleoside 1-alkynylphosphonates

  • Author/Authors

    Maïa Meurillon، نويسنده , , Franck Gallier، نويسنده , , Suzanne Peyrottes، نويسنده , , Christian Perigaud، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2009
  • Pages
    8
  • From page
    6039
  • To page
    6046
  • Abstract
    A series of ribonucleoside 1-alkynylphosphonates have been synthesized using a palladium-catalyzed phosphonylation of terminal 1,1-dibromo-1-alkene nucleosidic derivatives and high selectivity for product distribution was observed during this step. Both nucleosidic and osidic pathways were explored and the corresponding optimization study is reported herein.
  • Keywords
    Nucleotide analogue , 1-Alkynylphosphonate , Sugar phosphonate
  • Journal title
    Tetrahedron
  • Serial Year
    2009
  • Journal title
    Tetrahedron
  • Record number

    1097358