• Title of article

    Benzotriazole: an efficient ligand for the copper-catalyzed N-arylation of indoles

  • Author/Authors

    Akhilesh Kumar Verma، نويسنده , , Jaspal Singh، نويسنده , , Richard C. Larock، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2009
  • Pages
    6
  • From page
    8434
  • To page
    8439
  • Abstract
    A general, efficient, and inexpensive method for the N-arylation of indoles using a catalytic system derived from CuI and benzotriazole is reported. Selective mono N-arylation of indoles with ortho-dihaloarenes has also been successfully achieved in good yields using this protocol.
  • Keywords
    Benzotriazole , Dihalobenzene , Indole , CuI , N-arylation
  • Journal title
    Tetrahedron
  • Serial Year
    2009
  • Journal title
    Tetrahedron
  • Record number

    1097807