• Title of article

    De novo synthesis of teleocidin B analogs

  • Author/Authors

    Jun Pu، نويسنده , , Kangwen Deng، نويسنده , , John Butera، نويسنده , , Michael Chlenov، نويسنده , , Adam Gilbert، نويسنده , , Mike Kagan، نويسنده , , James Mattes، نويسنده , , Lynn Resnick، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    10
  • From page
    1963
  • To page
    1972
  • Abstract
    Teleocidin B analogs have been synthesized in 24 steps and 1.9% overall yield. The key steps include aromatic Claisen rearrangement, intramolecular Heck reaction of a tetra-substituted alkene, and ruthenium (II) catalyzed indole cyclization. Teleocidin and the new analogs promote cell spreading on fibroblast cells that were treated with amino-Nogo, an inhibitor of cell spreading.
  • Keywords
    intramolecular Heck reaction , Claisen rearrangement , Ruthenium catalyzed indole cyclization , Teleocidin B
  • Journal title
    Tetrahedron
  • Serial Year
    2010
  • Journal title
    Tetrahedron
  • Record number

    1100623