• Title of article

    Synthesis of pyrimido[6,1-a]isoquinolines via a one-pot, four-component reaction

  • Author/Authors

    Abdolali Alizadeh، نويسنده , , Atieh Rezvanian، نويسنده , , Log-Guan Zhu، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    4
  • From page
    6924
  • To page
    6927
  • Abstract
    An efficient one-pot synthesis of pyrimido[6,1-a]isoquinoline-1-carboxylate derivatives is described. This involves the four-component reaction between primary amines, alkyl acetoacetates, isoquinoline and trichloromethylchloroformate (diphosgene) under mild conditions at ambient temperature.
  • Keywords
    Trichloromethylchloroformate , Alkyl acetoacetates , enaminone , Pyrimido-isoquinoline , Four-component reaction
  • Journal title
    Tetrahedron
  • Serial Year
    2010
  • Journal title
    Tetrahedron
  • Record number

    1101219