• Title of article

    Facile Cu-free Sonogashira cross-coupling of nucleoside C-6 arylsulfonates with terminal alkynes

  • Author/Authors

    Felix N. Ngassa، نويسنده , , Jamie M. Gomez، نويسنده , , Brandon E. Haines، نويسنده , , Michael J. Ostach، نويسنده , , Jared W. Hector، نويسنده , , Lindsay J. Hoogenboom، نويسنده , , Chelsea E. Page، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2010
  • Pages
    8
  • From page
    7919
  • To page
    7926
  • Abstract
    The combination of PdCl2[CH3CN]2 with XPhos is an efficient catalytic system for the Sonogashira-type cross-coupling of 2′-deoxyguanosine O6-arylsulfonates with terminal alkynes. The reactions generally proceed under mild conditions requiring no Cu co-catalyst to give the corresponding C-6-alkynylated deoxynucleosides in moderate to good yields.
  • Journal title
    Tetrahedron
  • Serial Year
    2010
  • Journal title
    Tetrahedron
  • Record number

    1101329