Regioselective Halogenation of 6-Azaindoles: Efficient Synthesis of 3-Halo-2,3-disubstituted-6-azaindole Derivatives
Author/Authors :
Gallou، Fabrice نويسنده , , Reeves، Jonathan T. نويسنده , , Tan، Zhulin نويسنده , , Song، Jinhua J. نويسنده , , Yee، Nathan K. نويسنده , , Campbell، Scot نويسنده , , Jones، Paul-James نويسنده , , Senanayake، Chris H. نويسنده ,
Issue Information :
روزنامه با شماره پیاپی سال 2005
Pages :
-23
From page :
24
To page :
0
Abstract :
A mild and efficient synthesis of 3-halo-2-substituted-6azaindoles was developed by regioselective halogenation of 6-a7.aindole systems. The transformation was achieved with copper(ll) bromide in acetonitrile at room temperature.
Keywords :
regioselective halogenation of 6-azaindoles , pyrrolopyridine , copper (II) bromide
