Title of article :
Efficient synthesis of new 3-heteroaryl-1-functionalized 1H-indazoles
Author/Authors :
Alberto Fraile، نويسنده , , M. Rosario Mart?n، نويسنده , , José Luis Garc?a Ruano، نويسنده , , Juan Antonio D?az، نويسنده , , Esther Arranz-Plaza، نويسنده ,
Issue Information :
هفته نامه با شماره پیاپی سال 2011
Abstract :
The efficient synthesis of novel 3-heteroaryl N-1-functionalized indazoles, via palladium cross-coupling reactions of ethyl (3-iodo-1H-indazol-1-yl)acetate with 2- and 3-pyrrolylboronic acids, 2-, 4- and 5-thiazolylstannanes, and other heteroarylmetallated derivatives are reported.
Keywords :
1H-Indazoles , Cross-coupling , Thiazole , C–C coupled heterocycles , azoles
Journal title :
Tetrahedron
Journal title :
Tetrahedron
