• Title of article

    Synthesis of gemini triethylene-tetramine bridged bis-tridentate iron(III) chelators

  • Author/Authors

    David Rodriguez-Lucena، نويسنده , , Isabelle J. Schalk، نويسنده , , Gaëtan L.A. Mislin، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    6
  • From page
    2149
  • To page
    2154
  • Abstract
    Eight gemini bis-2-(2-hydroxyphenyl)-thiazole-4-carboxamide and -thiocarboxamide (BHPTC) chelators were efficiently synthesized. Mass spectrometry showed these compounds all form 1:1 complexes with iron(III). Three of these chelators exhibit promising antiproliferative activities when tested on human cancerous cell lines.
  • Keywords
    Cancer , Iron chelation therapy , Triethylene-tetramine , Iron chelator , BHPTC , Thioamide
  • Journal title
    Tetrahedron
  • Serial Year
    2011
  • Journal title
    Tetrahedron
  • Record number

    1103048