• Title of article

    Petasis Boronic Mannich Reactions of Electron-Poor Aromatic Amines under Microwave Conditions

  • Author/Authors

    Follmann، Markus نويسنده , , Graul، Franziska نويسنده , , Schafer، Thorsten نويسنده , , Kopec، Sebastian نويسنده , , Hamley، Peter نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2005
  • Pages
    -1008
  • From page
    1009
  • To page
    0
  • Abstract
    The Petasis reaction of electron-poor aromatic amines such as aminopyridines under microwave irradiation conditions is described. The process provides rapid access to a number of unnatural N-aryl-(alpha)-amino acids. The influence of the electronic demand of the boronic acids on the yields is discussed. A comparison with conventional heating is provided.
  • Keywords
    multicomponent reactions , amino acids , boron , Green chemistry , Heterocycles
  • Journal title
    Synlett
  • Serial Year
    2005
  • Journal title
    Synlett
  • Record number

    110313