• Title of article

    Direct annulation and alkylation of indoles with 2-aminobenzyl alcohols catalyzed by TFA

  • Author/Authors

    Forest J. Robertson، نويسنده , , Bradshaw D. Kenimer، نويسنده , , Jimmy Wu، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2011
  • Pages
    6
  • From page
    4327
  • To page
    4332
  • Abstract
    An efficient method for the annulation of indoles with 2-aminobenzyl alcohols, catalyzed by TFA, to furnish 5,6-fused indoline aminals is reported. This method can be extended to the alkylation of indoles at C3. 2-Aminobenzyl alcohols are used directly without recourse to protection of the aniline nitrogen or activation of the alcohol.
  • Keywords
    annulation , Alkylation , Indole , Alcohol , Communesin
  • Journal title
    Tetrahedron
  • Serial Year
    2011
  • Journal title
    Tetrahedron
  • Record number

    1103306

    • Link To Document
    https://search.isc.ac/dl/search/defaultta.aspx?DTC=10&DC=1103306