Title of article
A Versatile Synthesis of 7-Azaindoles
Author/Authors
Schirok، Hartmut نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2005
Pages
-1254
From page
1255
To page
0
Abstract
1,3-Disubstituted 7-azaindoles were synthesized from 2,6-dichloropyridine using DoM and intramolecular aromatic substitution after epoxide opening by an amine. Even the sterically demanding adamantylamine may be incorporated leading to derivatives which are not accessible by alkylation of the parent compound.
Keywords
pyridines , Metalations , nucleophilic aromatic substitutions , azaindoles , ring closure
Journal title
Synlett
Serial Year
2005
Journal title
Synlett
Record number
110411
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