• Title of article

    The acid-mediated ring opening/cyclisation reaction of N-benzyl-α-aryl-azetidinones

  • Author/Authors

    Frank D. King، نويسنده , , Stephen Caddick، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2012
  • Pages
    5
  • From page
    9350
  • To page
    9354
  • Abstract
    N-Benzyl-4-aryl-azetidinones undergo ring opening with triflic acid to form N-benzyl-cinnamamides, which either undergo cyclisation to give 5-aryl-benzazepin-3-ones or N-debenzylation to give cinnamamides.
  • Keywords
    Triflic acid , intramolecular cyclisation , Benzazepin-3-ones , azetidinone , cinnamamides
  • Journal title
    Tetrahedron
  • Serial Year
    2012
  • Journal title
    Tetrahedron
  • Record number

    1105113