• Title of article

    Diastereoselective and one-pot synthesis of trans-isoquinolonic acids via three-component condensation of homophthalic anhydride, aldehydes, and ammonium acetate catalyzed by aspartic acid

  • Author/Authors

    Arash Ghorbani-Choghamarani، نويسنده , , Maryam Hajjami، نويسنده , , Masoomeh Norouzi، نويسنده , , Yunes Abbasityula، نويسنده , , Vaclav Eigner، نويسنده , , Michal Dusek، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2013
  • Pages
    4
  • From page
    6541
  • To page
    6544
  • Abstract
    Aspartic acid has been developed as a versatile and highly efficient organocatalyst for the three component combination of homophthalic anhydride, aldehydes, and ammonium acetate to afford trans-isoquinolonic acids. The reactions were carried out in acetonitrile under reflux conditions. Aspartic acid as an efficient organocatalyst exhibits dramatically improved diastereoselectivity compared with previously reported catalysts for this synthetic strategy.
  • Keywords
    Isoquinolonic acid , Diastereoselective , Aldehyde , Homophthalic anhydride , ammonium acetate
  • Journal title
    Tetrahedron
  • Serial Year
    2013
  • Journal title
    Tetrahedron
  • Record number

    1106059