• Title of article

    A sort synthesis of polyhydroxylated pyrrolizidines via sequential 1,3-dipolar cycloaddition and reductive amination

  • Author/Authors

    Petros Gkizis، نويسنده , , Nikolaos G. Argyropoulos، نويسنده , , Evdoxia Coutouli-Argyropoulou، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2013
  • Pages
    8
  • From page
    8921
  • To page
    8928
  • Abstract
    Polyhydroxylated pyrrolizidines bearing a methyl group at C-5 have been synthesized by 1,3-dipolar cycloaddition of five membered cyclic nitrones with methyl vinyl ketone followed by a N–O reductive cleavage and in situ intramolecular reductive amination. The stereochemistry of the obtained compounds is examined in relation to the reactions mechanism.
  • Keywords
    Reductive amination , 1 , Azasugars , 3-dipolar cycloaddition , pyrrolizidines , Nitrones
  • Journal title
    Tetrahedron
  • Serial Year
    2013
  • Journal title
    Tetrahedron
  • Record number

    1106335