• Title of article

    Electrophilic Fluorination of 5-(Cyanomethyl)imidazole-4-carboxylate Nucleosides: Facile Entry to 3-Fluoro-3-deazaguanosine Analogues

  • Author/Authors

    Sakthivel، Kandasamy نويسنده , , Cook، P. Dan نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2005
  • Pages
    -1585
  • From page
    1586
  • To page
    0
  • Abstract
    A facile and efficient methodology is described for the synthesis of 3fluoro-3-deazaguanosines based on a novel electrophilic fluorination of 5(cyanomethyl)imidazole-4-carboxylate nucleosides. This general methodology can be readily applied to the synthesis of sugar-modified 3fluoro-3-deazaguanosine analogues.
  • Keywords
    nucleosides , 3-deazapurine , 3-deazaguanosine , fluorinated nucleosides , electrophilic fluorination
  • Journal title
    Synlett
  • Serial Year
    2005
  • Journal title
    Synlett
  • Record number

    110703