Title of article
Synthesis of Ring-A-Substituted Tryptophan by a Palladium-Catalyzed Heteroamiulation Reaction
Author/Authors
Zhu، Jieping نويسنده , , Jia، Yanxing نويسنده ,
Issue Information
روزنامه با شماره پیاپی سال 2005
Pages
-2468
From page
2469
To page
0
Abstract
Coupling of substituted o-iodoanilines with methyl (S)2-N-,N-di-tert-butoxycarbonyl-5-oxo-pentanoate, derived from glutamic acid, in DMF in the presence of palladium acetate and DABCO provides substituted tryptophans in good to excellent yields.
Keywords
palladium-catalyzed heteroannulation , substituted tryptophan , indole synthesis
Journal title
Synlett
Serial Year
2005
Journal title
Synlett
Record number
110836
Link To Document