• Title of article

    Synthesis of Ring-A-Substituted Tryptophan by a Palladium-Catalyzed Heteroamiulation Reaction

  • Author/Authors

    Zhu، Jieping نويسنده , , Jia، Yanxing نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2005
  • Pages
    -2468
  • From page
    2469
  • To page
    0
  • Abstract
    Coupling of substituted o-iodoanilines with methyl (S)2-N-,N-di-tert-butoxycarbonyl-5-oxo-pentanoate, derived from glutamic acid, in DMF in the presence of palladium acetate and DABCO provides substituted tryptophans in good to excellent yields.
  • Keywords
    palladium-catalyzed heteroannulation , substituted tryptophan , indole synthesis
  • Journal title
    Synlett
  • Serial Year
    2005
  • Journal title
    Synlett
  • Record number

    110836