• Title of article

    Pd-Catalyzed Cyclization of 1-Allyl-2-indolecarboxamides by Intramolecular Amidation of Unactivated Ethylenic Bond

  • Author/Authors

    Abbiati، Giorgio نويسنده , , Beccalli، Egle نويسنده , , Broggini، Gianluigi نويسنده , , Martinelli، Michela نويسنده , , Paladino، Giuseppe نويسنده ,

  • Pages
    -72
  • From page
    73
  • To page
    0
  • Abstract
    The intramolecular Pd(II)-mediated cyclization of 1-allyl-2-indolecarboxamides leads to pyrazino[1,2-a]indoles through the conversion of the olefinic C-H bond into a C-N bond by ­reaction with an amide group. When operating on the allylamide, a domino process was observed with a double C-H functionalization.
  • Keywords
    cyclizations , fused-ring systems , indoles , Palladium , domino reactions
  • Journal title
    Astroparticle Physics
  • Record number

    110896