• Title of article

    Enolate Conjugate Addition to Alkylidene Bis-Sulfoxides: Sphaeric Acid Synthesis and Absolute Configuration Determination

  • Author/Authors

    Brebion، Franck نويسنده , , Goddard، Jean-Philippe نويسنده , , Gomez، Catherine نويسنده , , Fensterbank، Louis نويسنده , , Malacria، Max نويسنده ,

  • Pages
    -712
  • From page
    713
  • To page
    0
  • Abstract
    The first stereoselective synthesis of sphaeric acid is described. The key step of this synthesis is an efficient ester enolate conjugate addition onto alkylidene bissulfoxides with good to high diastereoselectivity. Formation of sphaeric acid allowed the determination of its absolute configuration as 2R,3R.
  • Keywords
    enolate addition , alkylidene bis-sulfoxides , sphaeric acid , E/Z-enolate , succinic acid
  • Journal title
    Astroparticle Physics
  • Record number

    111071