• Title of article

    design and synthesis of a novel series of HIV-1 protease inhibitors Original Research Article

  • Author/Authors

    Eiji Takashiro، نويسنده , , Yuji Nakamura، نويسنده , , Shuichi Miyamoto، نويسنده , , Yuji Ozawa، نويسنده , , Akiko Sugiyama، نويسنده , , Katsumi Fujimoto، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 1999
  • Pages
    10
  • From page
    2105
  • To page
    2114
  • Abstract
    The synthesis and the SAR study of novel pseudo symmetric inhibitors of HIV-1 protease are described. Michael addition of amino acid derivatives to vinyl ketones was utilized to derive a potent (nM) series of HIV-1 protease inhibitors.
  • Journal title
    Bioorganic and Medicinal Chemistry
  • Serial Year
    1999
  • Journal title
    Bioorganic and Medicinal Chemistry
  • Record number

    1300540