• Title of article

    Design and synthesis of trans 2-(furan-2-yl)vinyl heteroaromatic iodides with antitumour activity Original Research Article

  • Author/Authors

    Cosimo Gianluca Fortuna، نويسنده , , Vincenza Barresi، نويسنده , , Giuliano Berellini، نويسنده , , Giuseppe Musumarra، نويسنده ,

  • Issue Information
    روزنامه با شماره پیاپی سال 2008
  • Pages
    10
  • From page
    4150
  • To page
    4159
  • Abstract
    A new molecular modelling approach based on physico-chemical and pharmacokinetic properties, called Volsurf plus, was used to design new heterocyclic compounds with antiproliferative activity. The synthesis and in vitro antitumour tests on a breast carcinoma cell line (MCF7) confirmed VOLSURF predicted activity values.
  • Keywords
    Gold , Asinex , Structure-based virtual screening , SARS-3CLpro inhibitor
  • Journal title
    Bioorganic and Medicinal Chemistry
  • Serial Year
    2008
  • Journal title
    Bioorganic and Medicinal Chemistry
  • Record number

    1304246