Author/Authors :
Chi، نويسنده , , Sung Min and Choi، نويسنده , , Joong-Kwon and Yum، نويسنده , , Eul Kgun and Chi، نويسنده , , Dae Yoon، نويسنده ,
Abstract :
Palladium-catalyzed functionalization at the 2-position of various 5- and 7-azaindoles was performed by Suzuki, Heck, and Stille reactions. The 2-substituted azaindoles were obtained with 5% Pd(OAc)2, LiCl, and KOAc in DMF at 110°C with moderate to high yields.