• Title of article

    Structure of argifin, a new chitinase inhibitor produced by Gliocladium sp.

  • Author/Authors

    Shiomi، نويسنده , , Kazuro and Arai، نويسنده , , Noriko and Iwai، نويسنده , , Yuzuru and Turberg، نويسنده , , Andreas and K?lbl، نويسنده , , Heinz and ?mura، نويسنده , , Satoshi، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    3
  • From page
    2141
  • To page
    2143
  • Abstract
    A new chitinase inhibitor, named argifin, was isolated from the cultured broth of a fungal strain Gliocladium sp. FTD-0668. Argifin was a water-soluble cyclic pentapeptide, and its structure was elucidated as cyclo(Nω-(N-methylcarbamoyl)-l-arginyl-N-methyl-l-phenylalanyl-β-l-aspartyl-β-l-aspartyl-d-alanyl). The IC50 value of argifin against blowfly (Lucilia cuprina) chitinase was 3.7 μM.
  • Keywords
    enzyme inhibitor , fungi , natural product , Peptide
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2000
  • Journal title
    Tetrahedron Letters
  • Record number

    1636657