Title of article
Preparation of 5-substituted 2-carboxyindoles on solid support
Author/Authors
Tois، نويسنده , , Jan and Franzén، نويسنده , , Robert and Aitio، نويسنده , , Olli and Huikko، نويسنده , , Katri and Taskinen، نويسنده , , Jyrki، نويسنده ,
Issue Information
هفته نامه با شماره پیاپی سال 2000
Pages
4
From page
2443
To page
2446
Abstract
The preparation of 5-substituted 2-carboxyindoles on solid support is reported. In the approach, the indole moiety is synthesized in solution phase, followed by nitro-group reduction, reductive amination and alkylation on solid support. The method provides a simple and convenient route for the preparation of 5-substituted 2-carboxyindoles with high purity and good yield.
Journal title
Tetrahedron Letters
Serial Year
2000
Journal title
Tetrahedron Letters
Record number
1636800
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