• Title of article

    Synthesis of 18R-hydroxy-epiallo-yohimbines from (−)-3-iso-19,20-dehydro-β-yohimbine: an enantiospecific route to deserpidine and reserpine analogues from secologanin

  • Author/Authors

    Binns، نويسنده , , Falmai and Brown، نويسنده , , Richard T and Dauda، نويسنده , , Bukar E.N، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    5
  • From page
    5631
  • To page
    5635
  • Abstract
    (−)-3-Iso-19,20-dehydro-β-yohimbine has been converted into epiallo-yohimbines and, via a novel regio- and stereoselective hydration, into the 18R-hydroxy derivative, an analogue of deserpidine. Its 11-methoxy derivative, also prepared from secologanin, is a potential precursor for a reserpine analogue.
  • Keywords
    Alkaloids , indole , stereoselection , terpene , Addition reaction , regioselection
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2000
  • Journal title
    Tetrahedron Letters
  • Record number

    1638265