• Title of article

    Novel and highly efficient DNA photocleavers: hydroperoxides of heterocyclic-fused naphthalimides

  • Author/Authors

    Yao، نويسنده , , Wei and Qian، نويسنده , , Xuhong and Hu، نويسنده , , Qingyan، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    5
  • From page
    7711
  • To page
    7715
  • Abstract
    A series of novel hydroperoxides of heterocyclic-fused naphthalimides were designed, synthesized and exhibited excellent DNA photonicking activities. Among these compounds, the benzothiophenonaphthalimide-type reagent proved to be the most efficient, it can induce single-strand nicks in duplex DNA at micromolar concentration upon illumination. The relationship between the molecular structure and cleaving activities was discussed.
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2000
  • Journal title
    Tetrahedron Letters
  • Record number

    1639140