• Title of article

    A novel synthesis of 4′-thionucleosides and a potential stereospecific route to pyrimidine nucleosides

  • Author/Authors

    Miller، نويسنده , , J.Allen and Pugh، نويسنده , , Ashley W and Ullah، نويسنده , , G.Mustafa and Gutteridge، نويسنده , , Clare، نويسنده ,

  • Issue Information
    هفته نامه با شماره پیاپی سال 2000
  • Pages
    7
  • From page
    10099
  • To page
    10105
  • Abstract
    Starting with the l-ascorbate derived epoxide 1, a di-t-butyl dithioacetal cyclisation route to 2′-deoxy-4′-thionucleosides has been developed. Based on an intermediate in this route, a novel and stereospecific route to α- or β-pyrimidine nucleosides has been conceived, but its implementation failed at a key ring-closure step.
  • Keywords
    Epoxide opening , 2?-deoxy-4?-thionucleoside synthesis , di-t-butyl dithioacetal cyclisation
  • Journal title
    Tetrahedron Letters
  • Serial Year
    2000
  • Journal title
    Tetrahedron Letters
  • Record number

    1640689